TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataKi: <0.150nMAssay Description:Binding affinity to ATR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPurchase
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataKi: 0.580nMAssay Description:Binding affinity to PARP1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to PARP1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataKi: <100nMAssay Description:Inhibition of DNA-PK (unknown origin) assessed as inhibition constant using Glu-Pro-Pro-Leu-Ser-Gln-Glu-Ala-Phe-Ala-Asp-Leu-Trp-Lys-Lys-Lys peptide a...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataKi: <100nMAssay Description:Inhibition of DNA-PK (unknown origin) assessed as inhibition constant using Glu-Pro-Pro-Leu-Ser-Gln-Glu-Ala-Phe-Ala-Asp-Leu-Trp-Lys-Lys-Lys peptide a...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.580nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 0.590nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of DNA-PK (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 0.780nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK using p53 as substrate incubated for 30 mins in presence of by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM in human MCF7 cells using etoposide as substrate incubated for 1 hr by Cell Western assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of ATM in human MCF7 cells using etoposide as substrate incubated for 1 hr by Cell Western assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of full-length human DNA-PK expressed in baculovirus expression system using p53 as substrate incubated for 1 hr in presence of ATP by ELI...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of full-length human DNA-PK expressed in baculovirus expression system using p53 as substrate incubated for 1 hr in presence of ATP by ELI...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of tracer 178 from N-terminal GST-fused human WEE1 (215 to 646 residues) expressed in baculovirus expression system preincubated for 5 m...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: <1nMAssay Description:Inhibition of N-terminal GST-tagged full-length recombinant human CHK1 expressed in baculovirus infected Sf9 insect cells using FAM-P10 peptide as su...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: <1nMAssay Description:Inhibition of CHK1 (unknown origin)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK using p53 as substrate incubated for 30 mins in presence of by HTRF assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of N-terminal GST-tagged wild-type WEE1 (215 to 646 residues) (unknown origin) expressed in Sf21 insect cells incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human DNA-PK using p53 as substrate incubated for 30 mins in presence of by HTRF assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Displacement of tracer 178 from WEE1 (unknown origin) incubated for 1 hr by Lantha Screen assayMore data for this Ligand-Target Pair
TargetATR-interacting protein/Serine/threonine-protein kinase ATR(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human FLAG-tagged ATR/c-Myc-tagged ATRIP expressed in mammalian expression system using p53 as substrate incubated for 2 hrs by fluores...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of N-terminal GST-tagged wild-type WEE1 (215 to 646 residues) (unknown origin) expressed in Sf21 insect cells incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
TargetATR-interacting protein/Serine/threonine-protein kinase ATR(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human FLAG-tagged ATR/c-Myc-tagged ATRIP expressed in mammalian expression system using p53 as substrate incubated for 2 hrs by fluores...More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human DNA-PK using p53 as substrate incubated for 30 mins in presence of by HTRF assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of tankyrase 2 (unknown origin) incubated for 1 hr by chemiluminescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Displacement of tracer 178 from WEE1 (unknown origin) incubated for 1 hr by Lantha Screen assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of WEE1 (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibition of PI3K-alpha (unknown origin) incubated for 40 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of tankyrase 2 (unknown origin) incubated for 1 hr by chemiluminescence based assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of ATR (unknown origin)-driven CHK1 phosphorylationMore data for this Ligand-Target Pair
Ligand InfoPurchase
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of CHK2 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Hubei Polytechnic University
Curated by ChEMBL
Hubei Polytechnic University
Curated by ChEMBL
Affinity DataIC50: 9.60nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair