TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 187nMAssay Description:Inhibition of human PI3Kalpha by Kinase-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 187nMAssay Description:Inhibition of human PI3Kalpha by Kinase-Glo assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 281nMAssay Description:Inhibition of human PI3Kgamma by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 363nMAssay Description:Inhibition of human PI3Kgamma by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 758nMAssay Description:Inhibition of human PI3Kdelta by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of human PI3Kbeta by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 973nMAssay Description:Inhibition of human PI3Kdelta by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Zhuhai Campus Of Zunyi Medical University
Curated by ChEMBL
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of human PI3Kbeta by ADP-Glo assayMore data for this Ligand-Target Pair