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Found 23 Enz. Inhib. hit(s) with all data for entry = 50016275
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593816(CHEMBL5191459)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
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TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593818(CHEMBL5175473)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593821(CHEMBL5191714)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593823(CHEMBL5175439)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593819(CHEMBL5173245)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593820(CHEMBL5193606)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593817(CHEMBL5202679)
Affinity DataIC50:  10nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593824(CHEMBL5169542)
Affinity DataIC50:  17nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593827(CHEMBL5196879)
Affinity DataIC50:  21nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593822(CHEMBL5186283)
Affinity DataIC50:  25nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593828(CHEMBL5204430)
Affinity DataIC50:  48nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593829(CHEMBL5184834)
Affinity DataIC50:  127nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593826(CHEMBL5187570)
Affinity DataIC50:  135nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  187nMAssay Description:Inhibition of human PI3Kalpha by Kinase-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPurchasePDB
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593816(CHEMBL5191459)
Affinity DataIC50:  187nMAssay Description:Inhibition of human PI3Kalpha by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593825(CHEMBL5182910)
Affinity DataIC50:  220nMAssay Description:Inhibition of human native full length DNA-PK by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593816(CHEMBL5191459)
Affinity DataIC50:  281nMAssay Description:Inhibition of human PI3Kgamma by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  363nMAssay Description:Inhibition of human PI3Kgamma by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPurchasePDB
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593816(CHEMBL5191459)
Affinity DataIC50:  758nMAssay Description:Inhibition of human PI3Kdelta by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50593816(CHEMBL5191459)
Affinity DataIC50:  830nMAssay Description:Inhibition of human PI3Kbeta by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  973nMAssay Description:Inhibition of human PI3Kdelta by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPurchasePDB
In DepthDetails PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of human PI3Kbeta by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPurchasePDB
In DepthDetails PubMed