TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 128nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 227nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 245nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 285nMAssay Description:Inhibition of PARP-1 derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 7.22E+3nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC derived from human HeLa cell nucleusMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: 4.21E+4nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Qingdao University Medical College
Curated by ChEMBL
Qingdao University Medical College
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair