Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50016226
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593342(CHEMBL5184354)
Affinity DataIC50:  24nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593328(CHEMBL5205360)
Affinity DataIC50:  24nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593331(CHEMBL5208153)
Affinity DataIC50:  40nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593334(CHEMBL5194403)
Affinity DataIC50:  41nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593339(CHEMBL5197796)
Affinity DataIC50:  42nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593335(CHEMBL5192165)
Affinity DataIC50:  75nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593330(CHEMBL5188937)
Affinity DataIC50:  170nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593338(CHEMBL5174696)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593333(CHEMBL5202378)
Affinity DataIC50:  250nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593322(CHEMBL5178011)
Affinity DataIC50:  310nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593326(CHEMBL5177951)
Affinity DataIC50:  480nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593341(CHEMBL5209002)
Affinity DataIC50:  640nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593340(CHEMBL5190853)
Affinity DataIC50:  640nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593337(CHEMBL5205347)
Affinity DataIC50:  810nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593325(CHEMBL5189187)
Affinity DataIC50:  940nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593336(CHEMBL5186754)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593332(CHEMBL1078237)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50400094(CHEMBL427092)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593323(CHEMBL5199345)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593329(CHEMBL5207932)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593327(CHEMBL5188651)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50593324(CHEMBL5188998)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of HIF-1alpha (unknown origin) transcriptional activity expressed in HEK293T cells co-transfected with renilla and HRE-firelfly luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed