Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 5869
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98008(US8481743, 4)
Affinity DataKi:  19.2nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98007(US8481743, 3)
Affinity DataKi:  36.1nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98009(US8481743, 1)
Affinity DataKi:  82.8nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98006(US8481743, 2)
Affinity DataKi:  331nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98006(US8481743, 2)
Affinity DataKi:  4.40E+3nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98008(US8481743, 4)
Affinity DataKi: >2.00E+4nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98009(US8481743, 1)
Affinity DataKi: >2.00E+4nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM98007(US8481743, 3)
Affinity DataKi: >2.00E+4nMpH: 7.4Assay Description:Radioligand binding assay (for screening and dose-displacement) using u-opioid and ORL-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent