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Found 9 Enz. Inhib. hit(s) with all data for entry = 6937
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160576(US9045389, 8)
Affinity DataKi:  33nM ΔG°:  -39.7kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160577(US9045389, 9)
Affinity DataKi:  38nM ΔG°:  -39.4kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160575(US9045389, 7)
Affinity DataKi:  45nM ΔG°:  -39.0kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160583(US9045389, 18)
Affinity DataKi:  60nM ΔG°:  -38.3kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160578(US9045389, 10)
Affinity DataKi:  120nM ΔG°:  -36.7kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160580(US9045389, 12)
Affinity DataKi:  240nM ΔG°:  -35.1kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160579(US9045389, 11)
Affinity DataKi:  240nM ΔG°:  -35.1kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160581(US9045389, 13)
Affinity DataKi:  270nM ΔG°:  -34.9kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160582(US9045389, 14)
Affinity DataKi:  770nM ΔG°:  -32.4kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
In DepthDetails US Patent