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Found 11 Enz. Inhib. hit(s) with all data for entry = 6956
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161383(US9108956, 7)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161384(US9108956, 10 | US9108956, 11 | US9108956, 8 | US9...)
Affinity DataIC50:  130nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161377(US9108956, 1 | US9108956, 2 | US9108956, 3 | US910...)
Affinity DataIC50:  300nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161382(US9108956, 6)
Affinity DataIC50:  310nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161384(US9108956, 10 | US9108956, 11 | US9108956, 8 | US9...)
Affinity DataIC50:  570nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161384(US9108956, 10 | US9108956, 11 | US9108956, 8 | US9...)
Affinity DataIC50:  760nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161377(US9108956, 1 | US9108956, 2 | US9108956, 3 | US910...)
Affinity DataIC50:  820nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161384(US9108956, 10 | US9108956, 11 | US9108956, 8 | US9...)
Affinity DataIC50:  1.20E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161377(US9108956, 1 | US9108956, 2 | US9108956, 3 | US910...)
Affinity DataIC50:  1.40E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161377(US9108956, 1 | US9108956, 2 | US9108956, 3 | US910...)
Affinity DataIC50:  2.60E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM161377(US9108956, 1 | US9108956, 2 | US9108956, 3 | US910...)
Affinity DataIC50:  5.90E+3nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent