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Found 41 Enz. Inhib. hit(s) with all data for entry = 7172
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179530(US9126976, 61)
Affinity DataIC50:  7.5nMAssay Description:An in vitro assay for determining ICso's to identify compounds that inhibit CETP transfer activity is performed based on a modification of a publishe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179535(US9126976, 66)
Affinity DataIC50:  8nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179525(US9126976, 56)
Affinity DataIC50:  11nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179501(US9126976, 32)
Affinity DataIC50:  12nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179526(US9126976, 57)
Affinity DataIC50:  12nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179529(US9126976, 60)
Affinity DataIC50:  14nMAssay Description:An in vitro assay for determining ICso's to identify compounds that inhibit CETP transfer activity is performed based on a modification of a publishe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179527(US9126976, 58)
Affinity DataIC50:  16nMAssay Description:An in vitro assay for determining ICso's to identify compounds that inhibit CETP transfer activity is performed based on a modification of a publishe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179533(US9126976, 64)
Affinity DataIC50:  16nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179518(US9126976, 49)
Affinity DataIC50:  20nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179528(US9126976, 59)
Affinity DataIC50:  24nMAssay Description:An in vitro assay for determining ICso's to identify compounds that inhibit CETP transfer activity is performed based on a modification of a publishe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179537(US9126976, 68)
Affinity DataIC50:  25nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179536(US9126976, 67)
Affinity DataIC50:  29nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179511(US9126976, 42)
Affinity DataIC50:  45.1nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179510(US9126976, 41)
Affinity DataIC50:  45.2nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179522(US9126976, 53)
Affinity DataIC50:  56nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179509(US9126976, 40)
Affinity DataIC50:  57.1nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179505(US9126976, 36)
Affinity DataIC50:  67nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179523(US9126976, 54)
Affinity DataIC50:  69nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179498(US9126976, 29)
Affinity DataIC50:  105nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179534(US9126976, 65)
Affinity DataIC50:  157nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179538(US9126976, 69)
Affinity DataIC50:  163nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179503(US9126976, 34)
Affinity DataIC50:  169nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179519(US9126976, 50)
Affinity DataIC50:  193nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179520(US9126976, 51)
Affinity DataIC50:  209nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179515(US9126976, 46)
Affinity DataIC50:  210nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179512(US9126976, 43)
Affinity DataIC50:  270nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179517(US9126976, 48)
Affinity DataIC50:  310nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179531(US9126976, 62)
Affinity DataIC50:  326nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179502(US9126976, 33)
Affinity DataIC50:  428nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179513(US9126976, 44)
Affinity DataIC50:  460nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179507(US9126976, 38)
Affinity DataIC50:  461nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179508(US9126976, 39)
Affinity DataIC50:  548nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179516(US9126976, 47)
Affinity DataIC50:  630nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179521(US9126976, 52)
Affinity DataIC50:  682nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179514(US9126976, 45)
Affinity DataIC50:  750nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179504(US9126976, 35)
Affinity DataIC50:  1.16E+3nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179506(US9126976, 37)
Affinity DataIC50:  1.27E+3nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179499(US9126976, 30)
Affinity DataIC50:  1.40E+3nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179524(US9126976, 55)
Affinity DataIC50:  1.43E+3nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179532(US9126976, 63)
Affinity DataIC50:  1.57E+3nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM179500(US9126976, 31)
Affinity DataIC50:  2.76E+3nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent