Reaction Details Report a problem with these data
Target
Zinc finger protein mex-5
Ligand
BDBM53160
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM53160
Synonyms:
3-[2-(2-carboxyethyl)-5-phenyl-1-pyrrolyl]benzoic acid | 3-[2-(2-carboxyethyl)-5-phenyl-1H-pyrrol-1-yl]benzoic acid | 3-[2-(2-carboxyethyl)-5-phenyl-pyrrol-1-yl]benzoic acid | 3-[2-(2-carboxyethyl)-5-phenylpyrrol-1-yl]benzoic acid | 3-[2-(3-hydroxy-3-oxopropyl)-5-phenyl-pyrrol-1-yl]benzoic acid | MLS001195956 | SMR000558717 | cid_954366
Type:
Small organic molecule
Emp. Form.:
C20H17NO4
Mol. Mass.:
335.3533
SMILES:
OC(=O)CCc1ccc(-c2ccccc2)n1-c1cccc(c1)C(O)=O
Structure:
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