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Target
Tropomyosin alpha-1 chain
Ligand
BDBM79658
Substrate
n/a
Meas. Tech.
Fluorescence-based biochemical high throughput dose response assay for activators of the calcium sensitivity of cardiac Regulated Thin Filaments (RTF)
EC50
>71481±n/a nM
Citation
 PubChem, PC Fluorescence-based biochemical high throughput dose response assay for activators of the calcium sensitivity of cardiac Regulated Thin Filaments (RTF) PubChem Bioassay (2011)[AID] 
Target
Name:
Tropomyosin alpha-1 chain
Synonyms:
TPM1 | TPM1_PIG | cardiac alpha tropomyosin
Type:
Enzyme Catalytic Domain
Mol. Mass.:
32681.01
Organism:
Sus scrofa
Description:
P42639
Residue:
284
Sequence:
MDAIKKKMQMLKLDKENALDRAEQAEADKKAAEDRSKRLEDELVSLQKKLKATEDELDKYSEAPKDAQEKLELAEKKATDAEADVASLNRRIQLVEEELDRAQERLATALQKLEEAEKAADESERGMKVIESRAQKDEEKMEIQEIQLKEAKHIAEDADRKYEEVARKLVIIESDLERAEERAELSEGKCAELEEELKTVTNNLKSLEAQAEKYSQKEDKYEEEIKVLSDKLKEAETRAEFAERSVTKLEKSIDDLEDELYAQKLKYKAISEELDHALNDMTSI
  
Inhibitor
Name:
BDBM79658
Synonyms:
2,3-Dihydro-1H-cyclopenta[b]quinoxaline 4,9-dioxide | 9-oxidanidyl-2,3-dihydro-1H-cyclopenta[b]quinoxalin-4-ium 4-oxide | 9-oxido-2,3-dihydro-1H-cyclopenta[b]quinoxalin-4-ium 4-oxide | MLS000523724 | SMR000122797 | cid_327035
Type:
Small organic molecule
Emp. Form.:
C11H10N2O2
Mol. Mass.:
202.2093
SMILES:
[O-]N1C2=C(CCC2)[N+](=O)c2ccccc12 |t:2|
Structure:
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