Reaction Details
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Target
STE20/SPS1-related proline-alanine-rich protein kinase
Ligand
BDBM50267896
Substrate
n/a
Meas. Tech.
ChEMBL_1704121 (CHEMBL4055354)
IC50
3900±n/a nM
Citation
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More Info.:
Target
Name:
STE20/SPS1-related proline-alanine-rich protein kinase
Synonyms:
2.7.11.1 | PS/TK | PSTK1 | Pancreatic serine/threonine-protein kinase | Pask | STE20/SPS1-related proline-alanine-rich protein kinase | STK39_RAT | Serine/threonine-protein kinase 39 | Spak | Ste-20-related kinase | Stk39
Type:
PROTEIN
Mol. Mass.:
60047.97
Organism:
Rattus norvegicus
Description:
ChEMBL_117413
Residue:
553
Sequence:
MAEPSGSPVHVQLPQQAAPVTAAAAAPAAATSAPAPAPAPAAPAAPAPAPAAAPAPAPAAQAVGWPICRDAYELQEVIGSGATAVVQAALCKPRQERVAIKRINLEKCQTSMDELLKEIQAMSQCSHPNVVTYYTSFVVKDELWLVMKLLSGGSMLDIIKYIVNRGEHKNGVLEEAIIATILKEVLEGLDYLHRNGQIHRDLKAGNILLGEDGSVQIADFGVSAFLATGGDVTRNKVRKTFVGTPCWMAPEVMEQVRGYDFKADMWSFGITAIELATGAAPYHKYPPMKVLMLTLQNDPPTLETGVEDKEMMKKYGKSFRKLLSLCLQKDPSKRPTAAELLKCKFFQKAKNREYLIEKLLTRTPDIAQRAKKVRRVPGSSGHLHKTEDGDWEWSDDEMDEKSEEGKAAASQEKSRRVKEENPEISVNAGGIPEQIQSLSVHDSQGQPNANEDYREGPCAVNLVLRLRNSRKELNDIRFEFTPGRDTADGVSQELFSAGLVDGHDVVIVAANLQKIVDDPKALKTLTFKLASGCDGAEIPDEVKLIGFAQLSVS