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Target
Opioid receptor delta 1
Ligand
BDBM50001031
Substrate
n/a
Meas. Tech.
ChEMBL_1762418 (CHEMBL4197665)
Ki
5.5±n/a nM
Citation
 Turnaturi, R; Marrazzo, A; Parenti, C; Pasquinucci, L Benzomorphan scaffold for opioid analgesics and pharmacological tools development: A comprehensive review. Eur J Med Chem 148:410-422 (2018) [PubMed]  Article 
Target
Name:
Opioid receptor delta 1
Synonyms:
G_PROTEIN_RECEP_F1_2 domain-containing protein | OPRD1
Type:
PROTEIN
Mol. Mass.:
40412.11
Organism:
Macaca mulatta
Description:
ChEMBL_117789
Residue:
372
Sequence:
MEPAPSAGAALQPPLFANASDAYPSAFPNAGANASGPPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMKTWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGIGVPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTACTPSDGPGGGAAA
  
Inhibitor
Name:
BDBM50001031
Synonyms:
3-Allyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocin-8-ol | CHEMBL330376 | SKF 10,047 (+) | SKF 10,047 (-) | SKF 10047
Type:
Small organic molecule
Emp. Form.:
C17H23NO
Mol. Mass.:
257.3706
SMILES:
C[C@H]1[C@H]2Cc3ccc(O)cc3[C@@]1(C)CCN2CC=C |TLB:16:15:1:10.4.3|
Structure:
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