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Target
Testis-specific serine/threonine-protein kinase 3
Ligand
BDBM50505541
Substrate
n/a
Meas. Tech.
ChEMBL_1823100 (CHEMBL4322864)
Kd
380±n/a nM
Citation
Hirozane, Y; Toyofuku, M; Yogo, T; Tanaka, Y; Sameshima, T; Miyahisa, I; Yoshikawa, M Structure-based rational design of staurosporine-based fluorescent probe with broad-ranging kinase affinity for kinase panel application. Bioorg Med Chem Lett 29:0 (2019) [PubMed] Article
More Info.:
Target
Name:
Testis-specific serine/threonine-protein kinase 3
Synonyms:
SPOGA3 | SPOGA3 | STK22C | Serine/threonine-protein kinase 22C | TSK-3 | TSSK-3 | TSSK3 | TSSK3_HUMAN | Testis-specific kinase 3 | Testis-specific serine/threonine-protein kinase 3
Type:
PROTEIN
Mol. Mass.:
30102.61
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109599
Residue:
268
Sequence:
MEDFLLSNGYQLGKTIGEGTYSKVKEAFSKKHQRKVAIKVIDKMGGPEEFIQRFLPRELQIVRTLDHKNIIQVYEMLESADGKICLVMELAEGGDVFDCVLNGGPLPESRAKALFRQMVEAIRYCHGCGVAHRDLKCENALLQGFNLKLTDFGFAKVLPKSHRELSQTFCGSTAYAAPEVLQGIPHDSKKGDVWSMGVVLYVMLCASLPFDDTDIPKMLWQQQKGVSFPTHLSISADCQDLLKRLLEPDMILRPSIEEVSWHPWLAST