Reaction Details Report a problem with these data
Target
Apelin receptor
Ligand
BDBM50583278
Substrate
n/a
Meas. Tech.
ChEMBL_2156909 (CHEMBL5041569)
Ki
>10000±n/a nM
Citation
Tran, K; Sainsily, X; Côté, J; Coquerel, D; Couvineau, P; Saibi, S; Haroune, L; Besserer-Offroy, É; Flynn-Robitaille, J; Resua Rojas, M; Murza, A; Longpré, JM; Auger-Messier, M; Lesur, O; Bouvier, M; Marsault, É; Boudreault, PL; Sarret, P Size-Reduced Macrocyclic Analogues of [Pyr J Med Chem 65:531-551 (2022) [PubMed] Article
More Info.:
Target
Name:
Apelin receptor
Synonyms:
AGTRL1 | APJ | APJ_HUMAN | APLNR | Angiotensin receptor-like 1 | Apelin receptor | Apelin receptor (APJ) | G-protein coupled receptor APJ | G-protein coupled receptor HG11
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42664.06
Organism:
Homo sapiens (Human)
Description:
P35414
Residue:
380
Sequence:
MEEGGDFDNYYGADNQSECEYTDWKSSGALIPAIYMLVFLLGTTGNGLVLWTVFRSSREKRRSADIFIASLAVADLTFVVTLPLWATYTYRDYDWPFGTFFCKLSSYLIFVNMYASVFCLTGLSFDRYLAIVRPVANARLRLRVSGAVATAVLWVLAALLAMPVMVLRTTGDLENTTKVQCYMDYSMVATVSSEWAWEVGLGVSSTTVGFVVPFTIMLTCYFFIAQTIAGHFRKERIEGLRKRRRLLSIIVVLVVTFALCWMPYHLVKTLYMLGSLLHWPCDFDLFLMNIFPYCTCISYVNSCLNPFLYAFFDPRFRQACTSMLCCGQSRCAGTSHSSSGEKSASYSSGHSQGPGPNMGKGGEQMHEKSIPYSQETLVVD