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Target
X-box-binding protein 1
Ligand
BDBM68010
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
10000±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM68010
Synonyms:
(2Z,6E)-4-tert-butyl-2,6-bis(2-furanylmethylidene)-1-cyclohexanone | (2Z,6E)-4-tert-butyl-2,6-bis(2-furfurylidene)cyclohexanone | (2Z,6E)-4-tert-butyl-2,6-bis(2-furylmethylene)cyclohexanone | (2Z,6E)-4-tert-butyl-2,6-bis(furan-2-ylmethylidene)cyclohexan-1-one | MLS000580624 | SMR000204787 | cid_12004979
Type:
Small organic molecule
Emp. Form.:
C20H22O3
Mol. Mass.:
310.3869
SMILES:
CC(C)(C)C1C\C(=C\c2ccco2)C(=O)\C(C1)=C\c1ccco1
Structure:
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