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Target
Lymphocyte antigen 6K
Ligand
BDBM50406016
Substrate
n/a
Meas. Tech.
ChEMBL_2266123
Kd
300±n/a nM
Citation
 Prakash, R; Goodlett, DW; Varghese, S; Andrys, J; Gbadamosi, FA; Arriaza, RH; Patel, M; Tiwari, PB; Borowski, T; Chruszcz, M; Shimizu, LS; Upadhyay, G Development of fluorophore labeled or biotinylated anticancer small molecule NSC243928. Bioorg Med Chem 79:0 (2023) [PubMed] 
Target
Name:
Lymphocyte antigen 6K
Synonyms:
LY6K | Ly-6K | Lymphocyte antigen 6K | Synonyms=CO16
Type:
PROTEIN
Mol. Mass.:
18674.17
Organism:
Homo sapiens
Description:
ChEMBL_120883
Residue:
165
Sequence:
MALLALLLVVALPRVWTDANLTARQRDPEDSQRTDEGDNRVWCHVCERENTFECQNPRRCKWTEPYCVIAAVKIFPRFFMVAKQCSAGCAAMERPKPEEKRFLLEEPMPFFYLKCCKIRYCNLEGPPINSSVFKEYAGSMGESCGGLWLAILLLLASIAAGLSLS
  
Inhibitor
Name:
BDBM50406016
Synonyms:
CHEMBL5281008
Type:
Small organic molecule
Emp. Form.:
C49H69N7O13S2
Mol. Mass.:
1028.241
SMILES:
[H][C@]12CS[C@@H](CCCCC(=O)NCCOCCOCCOCCOCCOCCOCCOCCNC(=O)c3ccc4c(Nc5ccc(NS(=O)(=O)CC)cc5OC)c5ccccc5nc4c3)[C@@]1([H])NC(=O)N2 |r|
Structure:
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