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Target
Phospholipase A2, membrane associated
Ligand
BDBM50274442
Substrate
n/a
Meas. Tech.
ChEMBL_537136 (CHEMBL989796)
IC50
>1600±n/a nM
Citation
 Oslund, RC; Cermak, N; Verlinde, CL; Gelb, MH Simplified YM-26734 inhibitors of secreted phospholipase A2 group IIA. Bioorg Med Chem Lett 18:5415-9 (2008) [PubMed]  Article 
Target
Name:
Phospholipase A2, membrane associated
Synonyms:
PA2GA_MOUSE | Pla2g2a
Type:
PROTEIN
Mol. Mass.:
16162.44
Organism:
Mus musculus
Description:
ChEMBL_352635
Residue:
146
Sequence:
MKVLLLLAASIMAFGSIQVQGNIAQFGEMIRLKTGKRAELSYAFYGCHCGLGGKGSPKDATDRCCVTHDCCYKSLEKSGCGTKLLKYKYSHQGGQITCSANQNSCQKRLCQCDKAAAECFARNKKTYSLKYQFYPNMFCKGKKPKC
  
Inhibitor
Name:
BDBM50274442
Synonyms:
1-(3-Dodecanoyl-2-hydroxy-5-methyl-phenyl)-dodecan-1-one | CHEMBL484180
Type:
Small organic molecule
Emp. Form.:
C31H52O3
Mol. Mass.:
472.7428
SMILES:
CCCCCCCCCCCC(=O)c1cc(C)cc(C(=O)CCCCCCCCCCC)c1O
Structure:
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