Reaction Details
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Target
5-hydroxytryptamine receptor 6
Ligand
BDBM50240514
Substrate
n/a
Meas. Tech.
ChEMBL_3664 (CHEMBL620800)
Ki
3±n/a nM
Citation
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More Info.:
Target
Name:
5-hydroxytryptamine receptor 6
Synonyms:
5-HT-6 | 5-HT6 | 5-hydroxytryptamine receptor 6 (5-HT-6) | 5-hydroxytryptamine receptor 6 (5-HT6R) | 5-hydroxytryptamine receptor 6 (5HT6) | 5HT6R_HUMAN | HTR6 | Serotonin (5-HT3) receptor | Serotonin 6 (5-HT6) receptor | Serotonin Receptor 6
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
46968.43
Organism:
Homo sapiens (Human)
Description:
P50406
Residue:
440
Sequence:
MVPEPGPTANSTPAWGAGPPSAPGGSGWVAAALCVVIALTAAANSLLIALICTQPALRNTSNFFLVSLFTSDLMVGLVVMPPAMLNALYGRWVLARGLCLLWTAFDVMCCSASILNLCLISLDRYLLILSPLRYKLRMTPLRALALVLGAWSLAALASFLPLLLGWHELGHARPPVPGQCRLLASLPFVLVASGLTFFLPSGAICFTYCRILLAARKQAVQVASLTTGMASQASETLQVPRTPRPGVESADSRRLATKHSRKALKASLTLGILLGMFFVTWLPFFVANIVQAVCDCISPGLFDVLTWLGYCNSTMNPIIYPLFMRDFKRALGRFLPCPRCPRERQASLASPSLRTSHSGPRPGLSLQQVLPLPLPPDSDSDSDAGSGGSSGLRLTAQLLLPGEATQDPPLPTRAAAAVNFFNIDPAEPELRPHPLGIPTN
Inhibitor
Name:
BDBM50240514
Synonyms:
(3Z)-3-(2-chloro-9H-thioxanthen-9-ylidene)-N,N-dimethylpropan-1-amine | (Z)-2-Chloro-9-(omega-dimethylaminopropylidene)thioxanthene | (Z)-chlorprothixene | CHEMBL908 | CHLORPROTHIXENE | cis-2-Chloro-9-(3-dimethylaminopropylidene)thioxanthene
Type:
Small organic molecule
Emp. Form.:
C18H18ClNS
Mol. Mass.:
315.86
SMILES:
CN(C)CC\C=C1\c2ccccc2Sc2ccc(Cl)cc12