Reaction Details
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Target
Histone-lysine N-methyltransferase KMT5C
Ligand
BDBM223980
Substrate
n/a
Meas. Tech.
Scintillation Proximity Assay (SPA)
pH
8±0
Temperature
298.15±0 K
IC50
1.2e+3±n/a nM
Citation
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More Info.:
Target
Name:
Histone-lysine N-methyltransferase KMT5C
Synonyms:
Histone-lysine N-methyltransferase SUV420H2 | KMT5C | KMT5C_HUMAN | Lysine N-methyltransferase 5C | Protein lysine methyltransferase SUV4-20H2 (SUV4-20H2) | SUV420H2 | Su(var)4-20 homolog 2 | Suppressor of variegation 4-20 homolog 2 | Suv4-20h2
Type:
Enzyme
Mol. Mass.:
52147.69
Organism:
Homo sapiens (Human)
Description:
Q86Y97
Residue:
462
Sequence:
MGPDRVTARELCENDDLATSLVLDPYLGFRTHKMNVSPVPPLRRQQHLRSALETFLRQRDLEAAYRALTLGGWTARYFQSRGPRQEAALKTHVYRYLRAFLPESGFTILPCTRYSMETNGAKIVSTRAWKKNEKLELLVGCIAELREADEGLLRAGENDFSIMYSTRKRSAQLWLGPAAFINHDCKPNCKFVPADGNAACVKVLRDIEPGDEVTCFYGEGFFGEKNEHCECHTCERKGEGAFRTRPREPALPPRPLDKYQLRETKRRLQQGLDSGSRQGLLGPRACVHPSPLRRDPFCAACQPLRLPACSARPDTSPLWLQWLPQPQPRVRPRKRRRPRPRRAPVLSTHHAARVSLHRWGGCGPHCRLRGEALVALGQPPHARWAPQQDWHWARRYGLPYVVRVDLRRLAPAPPATPAPAGTPGPILIPKQALAFAPFSPPKRLRLVVSHGSIDLDVGGEEL