Reaction Details Report a problem with these data
Target
Hemagglutinin
Ligand
BDBM525153
Substrate
n/a
Meas. Tech.
Cellular Assay-Influenza Virus Replication PR8 and X31 in Calu-3 Human Bronchial Epithelial Cells
EC50
34.0±n/a nM
Citation
Boudreault, P; Colombo, null; Leduc, R; Marsault, E; Plancq, B; Richter, M Matriptase inhibitors and uses thereof US Patent US10988505 Publication Date 4/27/2021
More Info.:
Target
Name:
Hemagglutinin
Synonyms:
HA | HEMA_I000X | Influenza A virus Hemagglutinin
Type:
PROTEIN
Mol. Mass.:
63574.85
Organism:
Influenza A virus (strain A/X-31 H3N2)
Description:
ChEMBL_884910
Residue:
566
Sequence:
MKTIIALSYIFCLALGQDLPGNDNSTATLCLGHHAVPNGTLVKTITDDQIEVTNATELVQSSSTGKICNNPHRILDGIDCTLIDALLGDPHCDVFQKETWDLFVERSKAFSNCYPYDVPDYASLRSLVASSGTLEFITEGFTWTGVTQNGGSIACKRGPDSGFFSRLNWLTKSESTYPVLNVTMPNNDNFDKLYIWGIHHPSTNQEQTSLYVQASGRVTVSTRRSQQTIIPNIGSRPWVRGLSSRISIYWTIVKPGDVLVINSNGNLIAPRGYFKMRTGKSSIMRSDAPIDTCISECITPNGSIPNDKPFQNVNKITYGACPKYVKQNTLKLATGMRNVPEKQTRGLFGAIAGFIENGWEGMIDGWYGFRHQNSEGTGQAADLKSTQAAIDQINGKLNRVIEKTNEKFHQIEKEFSEVEGRIQDLEKYVEDTKIDLWSYNAELLVALENQHTIDLTDSEMNKLFEKTRRQLRENAEDMGNGCFKIYHKCDNACIESIRNGTYDHDVYRDEALNNRFQIKGVELKSGYKDWILWISFAISCFLLCVVLLGFIMWTCQRGNIRCNICI