Reaction Details Report a problem with these data
Target
Complement factor D
Ligand
BDBM559426
Substrate
n/a
Meas. Tech.
Factor D Esterolytic Assay
IC50
<1000±n/a nM
Citation
Kotian, PL; Babu, YS; Zhang, W; Lu, P; Wu, M; Lv, W; Nguyen, TX; Dang, Z; Chintareddy, VR; Kumar, VS; Raman, K Substituted benzofuran, benzopyrrole, benzothiophene, and structurally related complement inhibitors US Patent US11370774 Publication Date 6/28/2022
More Info.:
Target
Name:
Complement factor D
Synonyms:
Adipsin | C3 convertase activator | CFAD_HUMAN | CFD | DF | PFD | Properdin factor D
Type:
Protein
Mol. Mass.:
27039.19
Organism:
Homo sapiens (Human)
Description:
P00746
Residue:
253
Sequence:
MHSWERLAVLVLLGAAACAAPPRGRILGGREAEAHARPYMASVQLNGAHLCGGVLVAEQWVLSAAHCLEDAADGKVQVLLGAHSLSQPEPSKRLYDVLRAVPHPDSQPDTIDHDLLLLQLSEKATLGPAVRPLPWQRVDRDVAPGTLCDVAGWGIVNHAGRRPDSLQHVLLPVLDRATCNRRTHHDGAITERLMCAESNRRDSCKGDSGGPLVCGGVLEGVVTSGSRVCGNRKKPGIYTRVASYAAWIDSVLA