Reaction Details Report a problem with these data
Target
Abscisic acid receptor PYL1/Protein phosphatase 2C 16
Ligand
BDBM313215
Substrate
n/a
Meas. Tech.
PP2C Activity Assay
IC50
97.0±n/a nM
Citation
Loiseleur, O; Wendeborn, SV; Cutler, SR 2-oxo-3,4-dihydroquinolin-6-yl sulphonamide CPDS and their use as plant growth regulators US Patent US10167261 Publication Date 1/1/2019
More Info.:
Target
Name:
Abscisic acid receptor PYL1/Protein phosphatase 2C 16
Synonyms:
PYR1-HAB1
Type:
Protein
Mol. Mass.:
n/a
Description:
n/a
Components:
This complex has 2 components.
Component 1
Name:
Protein phosphatase 2C 16
Synonyms:
AtP2C-HA | AtPP2C16 | HAB1 | P2C-HA | P2C16_ARATH | PP2C HAB1 | Protein HYPERSENSITIVE TO ABA 1 | Protein phosphatase 2C HAB1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
55716.72
Organism:
Arabidopsis thaliana (Mouse-ear cress)
Description:
n/a
Residue:
511
Sequence:
MEEMTPAVAMTLSLAANTMCESSPVEITQLKNVTDAADLLSDSENQSFCNGGTECTMEDVSELEEVGEQDLLKTLSDTRSGSSNVFDEDDVLSVVEDNSAVISEGLLVVDAGSELSLSNTAMEIDNGRVLATAIIVGESSIEQVPTAEVLIAGVNQDTNTSEVVIRLPDENSNHLVKGRSVYELDCIPLWGTVSIQGNRSEMEDAFAVSPHFLKLPIKMLMGDHEGMSPSLTHLTGHFFGVYDGHGGHKVADYCRDRLHFALAEEIERIKDELCKRNTGEGRQVQWDKVFTSCFLTVDGEIEGKIGRAVVGSSDKVLEAVASETVGSTAVVALVCSSHIVVSNCGDSRAVLFRGKEAMPLSVDHKPDREDEYARIENAGGKVIQWQGARVFGVLAMSRSIGDRYLKPYVIPEPEVTFMPRSREDECLILASDGLWDVMNNQEVCEIARRRILMWHKKNGAPPLAERGKGIDPACQAAADYLSMLALQKGSKDNISIIVIDLKAQRKFKTRT
Component 2
Name:
Abscisic acid receptor PYL1
Synonyms:
ABI1-binding protein 6 | PYL1 | PYL1_ARATH | PYR1-like protein 1 | RCAR12 | Regulatory components of ABA receptor 9
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25355.15
Organism:
Arabidopsis thaliana (Mouse-ear cress)
Description:
n/a
Residue:
221
Sequence:
MANSESSSSPVNEEENSQRISTLHHQTMPSDLTQDEFTQLSQSIAEFHTYQLGNGRCSSLLAQRIHAPPETVWSVVRRFDRPQIYKHFIKSCNVSEDFEMRVGCTRDVNVISGLPANTSRERLDLLDDDRRVTGFSITGGEHRLRNYKSVTTVHRFEKEEEEERIWTVVLESYVVDVPEGNSEEDTRLFADTVIRLNLQKLASITEAMNRNNNNNNSSQVR