Target

Ligand

Substrate

Meas. Tech.

Enzyme Inhibition Assay

Citation

 Jiaang, WT; Chen, YS; Hsu, T; Wu, SH; Chien, CH; Chang, CN; Chang, SP; Lee, SJ; Chen, X Novel isoindoline compounds for potent and selective inhibition of prolyl dipeptidase DPP8. Bioorg Med Chem Lett 15:687-91 (2005) [PubMed]  Article Copy BDB DOI

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Name:

Dipeptidyl peptidase 2

Synonyms:

DAP II | DPP2 | DPP2_HUMAN | DPP7 | Dipeptidyl aminopeptidase II | Dipeptidyl peptidase 2 (DPP II) | Dipeptidyl peptidase 2 (DPP2) | Dipeptidyl peptidase II (DDP-II) | Dipeptidyl peptidase II (DPP II) | Dipeptidyl peptidase II (DPP2) | Dipeptidyl peptidase II and dipeptidyl peptidase IV (DPP2 and DPP4) | QPP | carboxytripeptidase | dipeptidyl arylamidase II | dipeptidyl(amino)peptidase II | dipeptidylarylamidase

Type:

Protein

Mol. Mass.:

54339.29

Organism:

Homo sapiens (Human)

Description:

Q9UHL4

Residue:

492

Sequence:

MGSAPWAPVLLLALGLRGLQAGARRAPDPGFQERFFQQRLDHFNFERFGNKTFPQRFLVSDRFWVRGEGPIFFYTGNEGDVWAFANNSAFVAELAAERGALLVFAEHRYYGKSLPFGAQSTQRGHTELLTVEQALADFAELLRALRRDLGAQDAPAIAFGGSYGGMLSAYLRMKYPHLVAGALAASAPVLAVAGLGDSNQFFRDVTADFEGQSPKCTQGVREAFRQIKDLFLQGAYDTVRWEFGTCQPLSDEKDLTQLFMFARNAFTVLAMMDYPYPTDFLGPLPANPVKVGCDRLLSEAQRITGLRALAGLVYNASGSEHCYDIYRLYHSCADPTGCGTGPDARAWDYQACTEINLTFASNNVTDMFPDLPFTDELRQRYCLDTWGVWPRPDWLLTSFWGGDLRAASNIIFSNGNLDPWAGGGIRRNLSASVIAVTIQGGAHHLDLRASHPEDPASVVEARKLEATIIGEWVKAARREQQPALRGGPRLSL

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Name:

BDBM12195

Synonyms:

2-amino-4-{4-[bis(4-fluorophenyl)methyl]piperazin-1-yl}-1-(2,3-dihydro-1H-isoindol-2-yl)butane-1,4-dione | isoquinoline derivative 18

Type:

Small organic molecule

Emp. Form.:

C29H30F2N4O2

Mol. Mass.:

504.5709

SMILES:

NC(CC(=O)N1CCN(CC1)C(c1ccc(F)cc1)c1ccc(F)cc1)C(=O)N1Cc2ccccc2C1

Structure:

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Similarity to this molecule at least:

Name:

BDBM12196

Synonyms:

2,6-diamino-N-{1-[(4-nitrophenyl)carbamoyl]ethyl}hexanamide | Lys-Ala-p-nitroaniline | Lys-Ala-pNA

Type:

n/a

Emp. Form.:

n/a

Mol. Mass.:

n/a

SMILES:

n/a

Structure: