Reaction Details Report a problem with these data
Target
AP-4-A phosphorylase
Ligand
BDBM65570
Substrate
n/a
Meas. Tech.
FRET assay
pH
8±n/a
IC50
21800±3600 nM
Comments
extracted
Citation
Götz, KH; Hacker, SM; Mayer, D; Dürig, JN; Stenger, S; Marx, A Inhibitors of the Diadenosine Tetraphosphate Phosphorylase Rv2613c of Mycobacterium tuberculosis. ACS Chem Biol 12:2682-2689 (2017) [PubMed] Article
More Info.:
Target
Name:
AP-4-A phosphorylase
Synonyms:
AP,A phosphorylase | AP4A_MYCTU | ATP adenylyltransferase
Type:
Protein
Mol. Mass.:
21869.52
Organism:
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Description:
P9WMK9
Residue:
195
Sequence:
MSDEDRTDRATEDHTIFDRGVGQRDQLQRLWTPYRMNYLAEAPVKRDPNSSASPAQPFTEIPQLSDEEGLVVARGKLVYAVLNLYPYNPGHLMVVPYRRVSELEDLTDLESAELMAFTQKAIRVIKNVSRPHGFNVGLNLGTSAGGSLAEHLHVHVVPRWGGDANFITIIGGSKVIPQLLRDTRRLLATEWARQP