Reaction Details Report a problem with these data
Target
Proto-oncogene tyrosine-protein kinase receptor Ret [638-1114]
Ligand
BDBM296869
Substrate
n/a
Meas. Tech.
RET Kinase Enzymatic Assay
IC50
<10±n/a nM
Citation
Demartino, MP; Guan, HA Compounds as rearranged during transfection (RET) inhibitors US Patent US10292975 Publication Date 5/21/2019
More Info.:
Target
Name:
Proto-oncogene tyrosine-protein kinase receptor Ret [638-1114]
Synonyms:
CDHF12 | CDHR16 | PTC | Proto-oncogene tyrosine-protein kinase receptor Ret | RET | RET51 | RET_HUMAN
Type:
Protein
Mol. Mass.:
53601.71
Organism:
Homo sapiens (Human)
Description:
P07949[638-1114]
Residue:
477
Sequence:
IAAAVLFSFIVSVLLSAFCIHCYHKFAHKPPISSAEMTFRRPAQAFPVSYSSSGARRPSLDSMENQVSVDAFKILEDPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRKVGPGYLGSGGSRNSSSLDHPDERALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMVKRRDYLDLAASTPSDSLIYDDGLSEEETPLVDCNNAPLPRALPSTWIENKLYGMSDPNWPGESPVPLTRADGTNTGFPRYPNDSVYANWMLSPSAAKLMDTFDS