Reaction Details Report a problem with these data
Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43683
Substrate
n/a
Meas. Tech.
Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation
EC50
>55700±n/a nM
Citation
 PubChem, PC Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43683
Synonyms:
6-(1,3-benzoxazol-2-yl)-1,3-benzothiazol-2-amine | 6-Benzooxazol-2-yl-benzothiazol-2-ylamine | MLS000527641 | SMR000120215 | [6-(1,3-benzoxazol-2-yl)-1,3-benzothiazol-2-yl]amine | cid_810326
Type:
Small organic molecule
Emp. Form.:
C14H9N3OS
Mol. Mass.:
267.306
SMILES:
Nc1nc2ccc(cc2s1)-c1nc2ccccc2o1
Structure:
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