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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48118
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
6380±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48118
Synonyms:
3-(4-chlorophenyl)-6-(1-pyrrolidinyl)-1,2,4,5-tetrazine | 3-(4-chlorophenyl)-6-pyrrolidin-1-yl-1,2,4,5-tetrazine | 3-(4-chlorophenyl)-6-pyrrolidino-1,2,4,5-tetrazine | MLS000038815 | SMR000035727 | cid_535812
Type:
Small organic molecule
Emp. Form.:
C12H12ClN5
Mol. Mass.:
261.71
SMILES:
Clc1ccc(cc1)-c1nnc(nn1)N1CCCC1
Structure:
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