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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48145
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
9290±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48145
Synonyms:
3-methyl-N-(2-thiazolin-2-yl)coumarilamide | MLS000066288 | N-(4,5-dihydro-1,3-thiazol-2-yl)-3-methyl-1-benzofuran-2-carboxamide | N-(4,5-dihydrothiazol-2-yl)-3-methyl-2-benzofurancarboxamide | SMR000080715 | cid_1247112
Type:
Small organic molecule
Emp. Form.:
C13H12N2O2S
Mol. Mass.:
260.312
SMILES:
Cc1c(oc2ccccc12)C(=O)NC1=NCCS1 |t:15|
Structure:
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