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Target
D(1A) dopamine receptor
Ligand
BDBM40046
Substrate
n/a
Meas. Tech.
Allosteric Modulators of D1 Receptors: Dose-dependent Assay
EC50
0.0362±n/a nM
Citation
 PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Assay PubChem Bioassay (2007)[AID] 
Target
Name:
D(1A) dopamine receptor
Synonyms:
DA D1 receptor | DOPAMINE D1 | DRD1 | DRD1_HUMAN | Dopamine D1 receptor | Dopamine D1 receptor (D1R) | Dopamine D1A
Type:
Enzyme
Mol. Mass.:
49303.43
Organism:
Homo sapiens (Human)
Description:
P21728
Residue:
446
Sequence:
MRTLNTSAMDGTGLVVERDFSVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNATSLAETIDNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNCQTTTGNGKPVECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCGSGETQPFCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPATNNAIETVSINNNGAAMFSSHHEPRGSISKECNLVYLIPHAVGSSEDLKKEEAAGIARPLEKLSPALSVILDYDTDVSLEKIQPITQNGQHPT
  
Inhibitor
Name:
BDBM40046
Synonyms:
(4-methylbenzyl)-(tetrazolo[1,5-a]quinoxalin-4-yl)amine | MLS000091254 | N-(4-methylbenzyl)tetrazolo[1,5-a]quinoxalin-4-amine | N-[(4-methylphenyl)methyl]-4-tetrazolo[1,5-a]quinoxalinamine | N-[(4-methylphenyl)methyl]-[1,2,3,4]tetrazolo[1,5-a]quinoxalin-4-amine | N-[(4-methylphenyl)methyl]tetrazolo[1,5-a]quinoxalin-4-amine | SMR000025816 | cid_3243891
Type:
Small organic molecule
Emp. Form.:
C16H14N6
Mol. Mass.:
290.3226
SMILES:
Cc1ccc(CNc2nc3ccccc3n3nnnc23)cc1
Structure:
Search PDB for entries with ligand similarity: