Reaction Details Report a problem with these data
Target
Zinc finger protein mex-5
Ligand
BDBM52141
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52141
Synonyms:
2-[(1-oxo-2-phenoxyethyl)amino]propanoic acid [2-(2-benzofuranyl)-2-oxoethyl] ester | 2-[(2-phenoxyacetyl)amino]propionic acid [2-(benzofuran-2-yl)-2-keto-ethyl] ester | MLS000057997 | SMR000063043 | [2-(1-benzofuran-2-yl)-2-oxidanylidene-ethyl] 2-(2-phenoxyethanoylamino)propanoate | [2-(1-benzofuran-2-yl)-2-oxoethyl] 2-[(2-phenoxyacetyl)amino]propanoate | cid_2998385
Type:
Small organic molecule
Emp. Form.:
C21H19NO6
Mol. Mass.:
381.3787
SMILES:
CC(NC(=O)COc1ccccc1)C(=O)OCC(=O)c1cc2ccccc2o1
Structure:
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