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Target
Zinc finger protein mex-5
Ligand
BDBM52226
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52226
Synonyms:
2-(2,6-Dichloro-benzylsulfanyl)-N-(tetrahydro-furan-2-ylmethyl)-acetamide | 2-[(2,6-dichlorobenzyl)thio]-N-(tetrahydrofurfuryl)acetamide | 2-[(2,6-dichlorophenyl)methylsulfanyl]-N-(oxolan-2-ylmethyl)acetamide | 2-[(2,6-dichlorophenyl)methylthio]-N-(2-oxolanylmethyl)acetamide | 2-[[2,6-bis(chloranyl)phenyl]methylsulfanyl]-N-(oxolan-2-ylmethyl)ethanamide | MLS000122539 | SMR000119997 | cid_2947787
Type:
Small organic molecule
Emp. Form.:
C14H17Cl2NO2S
Mol. Mass.:
334.261
SMILES:
Clc1cccc(Cl)c1CSCC(=O)NCC1CCCO1
Structure:
Search PDB for entries with ligand similarity: