Reaction Details Report a problem with these data
Target
POsterior Segregation
Ligand
BDBM52074
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM52074
Synonyms:
3-Methoxy-N-{1-[4-(morpholine-4-sulfonyl)-phenyl]-piperidin-4-ylmethyl}-benzamide | 3-methoxy-N-[[1-(4-morpholin-4-ylsulfonylphenyl)piperidin-4-yl]methyl]benzamide | 3-methoxy-N-[[1-(4-morpholinosulfonylphenyl)-4-piperidyl]methyl]benzamide | 3-methoxy-N-[[1-[4-(4-morpholinylsulfonyl)phenyl]-4-piperidinyl]methyl]benzamide | MLS000068063 | SMR000000946 | cid_651404
Type:
Small organic molecule
Emp. Form.:
C24H31N3O5S
Mol. Mass.:
473.585
SMILES:
COc1cccc(c1)C(=O)NCC1CCN(CC1)c1ccc(cc1)S(=O)(=O)N1CCOCC1
Structure:
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