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Target
Kallikrein-5
Ligand
BDBM56146
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
50000±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Homo sapiens (Human)
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM56146
Synonyms:
2-[5-(1-azepanylsulfonyl)-4-chloro-2-methylphenoxy]acetamide | 2-[5-(azepan-1-ylsulfonyl)-4-chloranyl-2-methyl-phenoxy]ethanamide | 2-[5-(azepan-1-ylsulfonyl)-4-chloro-2-methyl-phenoxy]acetamide | 2-[5-(azepan-1-ylsulfonyl)-4-chloro-2-methylphenoxy]acetamide | MLS000049478 | SMR000075482 | cid_1288538
Type:
Small organic molecule
Emp. Form.:
C15H21ClN2O4S
Mol. Mass.:
360.856
SMILES:
Cc1cc(Cl)c(cc1OCC(N)=O)S(=O)(=O)N1CCCCCC1
Structure:
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