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Target
Kallikrein-5
Ligand
BDBM49905
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
50000±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Homo sapiens (Human)
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM49905
Synonyms:
2-(3-fluoranyl-4-methoxy-phenyl)-8-methyl-imidazo[1,2-a]pyridine | 2-(3-fluoro-4-methoxy-phenyl)-8-methyl-imidazo[1,2-a]pyridine | 2-(3-fluoro-4-methoxyphenyl)-8-methylimidazo[1,2-a]pyridine | MLS000688484 | SMR000284428 | cid_832352
Type:
Small organic molecule
Emp. Form.:
C15H13FN2O
Mol. Mass.:
256.2749
SMILES:
COc1ccc(cc1F)-c1cn2cccc(C)c2n1
Structure:
Search PDB for entries with ligand similarity: