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Target
Trans-activator protein BZLF1
Ligand
BDBM62417
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62417
Synonyms:
3-[[4-(dimethylsulfamoyl)benzoyl]amino]coumarilic acid ethyl ester | 3-[[[4-(dimethylsulfamoyl)phenyl]-oxomethyl]amino]-2-benzofurancarboxylic acid ethyl ester | MLS000093013 | SMR000028649 | cid_3238290 | ethyl 3-({4-[(dimethylamino)sulfonyl]benzoyl}amino)-1-benzofuran-2-carboxylate | ethyl 3-[[4-(dimethylsulfamoyl)benzoyl]amino]-1-benzofuran-2-carboxylate | ethyl 3-[[4-(dimethylsulfamoyl)phenyl]carbonylamino]-1-benzofuran-2-carboxylate
Type:
Small organic molecule
Emp. Form.:
C20H20N2O6S
Mol. Mass.:
416.448
SMILES:
CCOC(=O)c1oc2ccccc2c1NC(=O)c1ccc(cc1)S(=O)(=O)N(C)C
Structure:
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