Reaction Details
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X-box-binding protein 1
Ligand
BDBM34320
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
5370±n/a nM
Citation
More Info.:
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
Inhibitor
Name:
BDBM34320
Synonyms:
MLS000098038 | SMR000065677 | cid_2998049
Type:
Small organic molecule
Emp. Form.:
C21H25N5O
Mol. Mass.:
363.4561
SMILES:
CCCCC(CC)Cn1c2nc(C)oc(=N)c2c2nc3ccccc3nc12
Structure:
