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Target
X-box-binding protein 1
Ligand
BDBM54190
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
10000±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM54190
Synonyms:
1-[4-(difluoromethoxy)phenyl]-3-[3-(trifluoromethyl)phenyl]urea | 1-[4-[bis(fluoranyl)methoxy]phenyl]-3-[3-(trifluoromethyl)phenyl]urea | MLS000537683 | N-[4-(difluoromethoxy)phenyl]-N'-[3-(trifluoromethyl)phenyl]urea | SMR000143875 | cid_971803
Type:
Small organic molecule
Emp. Form.:
C15H11F5N2O2
Mol. Mass.:
346.2521
SMILES:
FC(F)Oc1ccc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc1
Structure:
Search PDB for entries with ligand similarity: