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Target
X-box-binding protein 1
Ligand
BDBM68080
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
2000±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM68080
Synonyms:
4,5-bis(bromanyl)-2-(4,6-dimethoxypyrimidin-2-yl)pyridazin-3-one | 4,5-dibromo-2-(4,6-dimethoxy-2-pyrimidinyl)-3(2H)-pyridazinone | 4,5-dibromo-2-(4,6-dimethoxy-2-pyrimidinyl)-3-pyridazinone | 4,5-dibromo-2-(4,6-dimethoxypyrimidin-2-yl)pyridazin-3-one | MLS000699101 | SMR000229896 | cid_985526
Type:
Small organic molecule
Emp. Form.:
C10H8Br2N4O3
Mol. Mass.:
392.004
SMILES:
COc1cc(OC)nc(n1)-n1ncc(Br)c(Br)c1=O
Structure:
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