Reaction Details Report a problem with these data
Target
Adenosine receptor A3
Ligand
BDBM81925
Substrate
n/a
Ki
2.9±n/a nM
Comments
PDSP_2952
Citation
Klotz, KN; Vogt, H; Tawfik-Schlieper, H Comparison of A1 adenosine receptors in brain from different species by radioligand binding and photoaffinity labelling. Naunyn Schmiedebergs Arch Pharmacol 343:196-201 (1991) [PubMed] Article
More Info.:
Target
Name:
Adenosine receptor A3
Synonyms:
AA3R_SHEEP | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADENOSINE A3 | ADORA1 | ADORA3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36152.74
Organism:
Sheep
Description:
ADENOSINE A1 ADORA1 Sheep::P35342
Residue:
317
Sequence:
MPVNSTAVSWTSVTYITVEILIGLCAIVGNVLVIWVVKLNPSLQTTTFYFIVSLALADIAVGVLVMPLAIVISLGVTIHFYSCLFMTCLMLIFTHASIMSLLAIAVDRYLRVKLTVRYRRVTTQRRIWLALGLCWLVSFLVGLTPMFGWNMKLSSADENLTFLPCRFRSVMRMDYMVYFSFFLWILVPLVVMCAIYFDIFYIIRNRLSQSFSGSRETGAFYGREFKTAKSLLLVLFLFALCWLPLSIINCILYFDGQVPQTVLYLGILLSHANSMMNPIVYAYKIKKFKETYLLILKACVMCQPSKSMDPSTEQTSE