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Target
D(2) dopamine receptor
Ligand
BDBM35256
Substrate
n/a
Ki
161±n/a nM
Comments
PDSP_1235
Citation
 Nicklaus, KJ; McGonigle, P; Molinoff, PB [3H]SCH 23390 labels both dopamine-1 and 5-hydroxytryptamine1c receptors in the choroid plexus. J Pharmacol Exp Ther 247:343-8 (1988) [PubMed] 
Target
Name:
D(2) dopamine receptor
Synonyms:
DOPAMINE D1 | DRD1 | DRD2 | DRD2_CANLF | Dopamine D2 receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
50587.58
Organism:
CANINE
Description:
DOPAMINE D1 DRD1 CANINE::Q9GJU1
Residue:
443
Sequence:
MDPLNLSWYDDDLESQNWSRPFNGSEGKPGKPHYNYYAMLLTLLIFIIVFGNVLVCMAVSREKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTASILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQNECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRRRRKRVNTERSSRAFRANLKAPLKGNCTHPEDMKLCTVIMKSNGSFPVNRRRVEAARRAQELEMEMLSSTSPPERTRYSPIPPSHHQLTLPDPSHHGLHSTADSPAKPEKNGHAKDHPKIAKIFEIQSMPNGKTRTSLKTMSRRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCECNIPPVLYSAFTWLGYVNSAVNPIIYTTFNIEFRKAFLKILHC
  
Inhibitor
Name:
BDBM35256
Synonyms:
(S)-mianserin | Lerivon | MIANSERIN | MIANSERIN (+) | MIANSERIN (-) | Tolvon
Type:
Small organic molecule
Emp. Form.:
C18H20N2
Mol. Mass.:
264.3648
SMILES:
[H][C@]12CN(C)CCN1c1ccccc1Cc1ccccc21 |r|
Structure:
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