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Target
Histamine H3 receptor
Ligand
BDBM50247053
Substrate
n/a
Meas. Tech.
ChEMBL_1712142 (CHEMBL4122191)
Ki
14±n/a nM
Citation
?a?ewska, D; Kaleta, M; Hagenow, S; Mogilski, S; Latacz, G; Karcz, T; Lubelska, A; Honkisz, E; Handzlik, J; Reiner, D; Sata?a, G; Filipek, B; Stark, H; Kie?-Kononowicz, K Novel naphthyloxy derivatives - Potent histamine H Bioorg Med Chem 26:2573-2585 (2018) [PubMed] Article
More Info.:
Target
Name:
Histamine H3 receptor
Synonyms:
HH3R | HRH3_MOUSE | Hrh3
Type:
PROTEIN
Mol. Mass.:
48560.37
Organism:
Mus musculus
Description:
ChEMBL_988451
Residue:
445
Sequence:
MERAPPDGLMNASGALAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFVADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCASSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAGPEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRYGVGEAGPGVETGEAGLGGGSGGGAAASPTSSSGSSSRGTERPRSLKRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGHCVPDYWYETSFWLLWANSAVNPVLYPLCHYSFRRAFTKLLCPQKLKVQPHGSLEQCWK