Reaction Details Report a problem with these data
Target
Solute carrier family 2, facilitated glucose transporter member 8
Ligand
BDBM50277370
Substrate
n/a
Meas. Tech.
ChEMBL_1717904 (CHEMBL4132904)
IC50
6000±n/a nM
Citation
Wei, C; Bajpai, R; Sharma, H; Heitmeier, M; Jain, AD; Matulis, SM; Nooka, AK; Mishra, RK; Hruz, PW; Schiltz, GE; Shanmugam, M Development of GLUT4-selective antagonists for multiple myeloma therapy. Eur J Med Chem 139:573-586 (2017) [PubMed] Article
More Info.:
Target
Name:
Solute carrier family 2, facilitated glucose transporter member 8
Synonyms:
GLUT-8 | GLUT8 | GLUTX1 | GTR8_HUMAN | Glucose transporter type 8 | Glucose transporter type X1 | SLC2A8 | Solute carrier family 2, facilitated glucose transporter member 8
Type:
PROTEIN
Mol. Mass.:
50822.02
Organism:
Homo sapiens
Description:
ChEMBL_118209
Residue:
477
Sequence:
MTPEDPEETQPLLGPPGGSAPRGRRVFLAAFAAALGPLSFGFALGYSSPAIPSLQRAAPPAPRLDDAAASWFGAVVTLGAAAGGVLGGWLVDRAGRKLSLLLCSVPFVAGFAVITAAQDVWMLLGGRLLTGLACGVASLVAPVYISEIAYPAVRGLLGSCVQLMVVVGILLAYLAGWVLEWRWLAVLGCVPPSLMLLLMCFMPETPRFLLTQHRRQEAMAALRFLWGSEQGWEDPPIGAEQSFHLALLRQPGIYKPFIIGVSLMAFQQLSGVNAVMFYAETIFEEAKFKDSSLASVVVGVIQVLFTAVAALIMDRAGRRLLLVLSGVVMVFSTSAFGAYFKLTQGGPGNSSHVAISAPVSAQPVDASVGLAWLAVGSMCLFIAGFAVGWGPIPWLLMSEIFPLHVKGVATGICVLTNWLMAFLVTKEFSSLMEVLRPYGAFWLASAFCIFSVLFTLFCVPETKGKTLEQITAHFEGR