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Target
Glycine receptor subunit alpha-3
Ligand
BDBM50229711
Substrate
n/a
Meas. Tech.
ChEMBL_1767509 (CHEMBL4219621)
EC50
454±n/a nM
Citation
Sparling, BA; DiMauro, EF Progress in the discovery of small molecule modulators of the Cys-loop superfamily receptors. Bioorg Med Chem Lett 27:3207-3218 (2017) [PubMed] Article
More Info.:
Target
Name:
Glycine receptor subunit alpha-3
Synonyms:
GLRA3 | GLRA3_HUMAN | Glycine receptor alpha-3/beta
Type:
PROTEIN
Mol. Mass.:
53809.29
Organism:
Homo sapiens (Human)
Description:
ChEMBL_967474
Residue:
464
Sequence:
MAHVRHFRTLVSGFYFWEAALLLSLVATKETDSARSRSAPMSPSDFLDKLMGRTSGYDARIRPNFKGPPVNVTCNIFINSFGSIAETTMDYRVNIFLRQKWNDPRLAYSEYPDDSLDLDPSMLDSIWKPDLFFANEKGANFHEVTTDNKLLRIFKNGNVLYSIRLTLTLSCPMDLKNFPMDVQTCIMQLESFGYTMNDLIFEWQDEAPVQVAEGLTLPQFLLKEEKDLRYCTKHYNTGKFTCIEVRFHLERQMGYYLIQMYIPSLLIVILSWVSFWINMDAAPARVALGITTVLTMTTQSSGSRASLPKVSYVKAIDIWMAVCLLFVFSALLEYAAVNFVSRQHKELLRFRRKRKNKTEAFALEKFYRFSDMDDEVRESRFSFTAYGMGPCLQAKDGMTPKGPNHPVQVMPKSPDEMRKVFIDRAKKIDTISRACFPLAFLIFNIFYWVIYKILRHEDIHQQQD