Reaction Details Report a problem with these data
Target
Peptidoglycan D,D-transpeptidase FtsI
Ligand
BDBM50378857
Substrate
n/a
Meas. Tech.
ChEMBL_553819 (CHEMBL966182)
IC50
187±n/a nM
Citation
More Info.:
Target
Name:
Peptidoglycan D,D-transpeptidase FtsI
Synonyms:
3.4.16.4 | AO964_07895 | CAZ03_05815 | CAZ10_21230 | CGU42_01090 | CRX60_22815 | CW299_32685 | DC19_24320 | DI492_11155 | DN070_30405 | DZ934_06595 | DZ940_08385 | DZ962_00565 | E4V10_06485 | EFK68_01815 | HQ52_24085 | IPC3_13380 | IPC669_10550 | NCTC13719_04773 | PAERUG_E15_London_28_01_14_00534 | PBP-3 | Penicillin-binding protein 3 | Peptidoglycan D,D-transpeptidase FtsI | RW109_RW109_05757 | ftsI_1 | ftsI_2 | pbpB
Type:
PROTEIN
Mol. Mass.:
62874.12
Organism:
Pseudomonas aeruginosa
Description:
ChEMBL_105732
Residue:
579
Sequence:
MKLNYFQGALYPWRFCVIVGLLLAMVGAIVWRIVDLHVIDHDFLKGQGDARSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKVSVGTKGYRENAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLPTATEQQQVNAAPAKGGRG