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Target
Protein ultraspiracle
Ligand
BDBM50488454
Substrate
n/a
Meas. Tech.
ChEMBL_925682 (CHEMBL3069808)
EC50
<50119±n/a nM
Citation
 Soin, T; Swevers, L; Kotzia, G; Iatrou, K; Janssen, CR; Rougé, P; Harada, T; Nakagawa, Y; Smagghe, G Comparison of the activity of non-steroidal ecdysone agonists between dipteran and lepidopteran insects, using cell-based EcR reporter assays. Pest Manag Sci 66:1215-29 (2010) [PubMed]  Article 
Target
Name:
Protein ultraspiracle
Synonyms:
Cf1 | Chorion factor 1 | NR2B4 | Nuclear receptor subfamily 2 group B member 4 | USP_DROME | XR2C | usp
Type:
PROTEIN
Mol. Mass.:
55254.53
Organism:
Drosophila melanogaster
Description:
ChEMBL_106725
Residue:
508
Sequence:
MDNCDQDASFRLSHIKEEVKPDISQLNDSNNSSFSPKAESPVPFMQAMSMVHVLPGSNSASSNNNSAGDAQMAQAPNSAGGSAAAAVQQQYPPNHPLSGSKHLCSICGDRASGKHYGVYSCEGCKGFFKRTVRKDLTYACRENRNCIIDKRQRNRCQYCRYQKCLTCGMKREAVQEERQRGARNAAGRLSASGGGSSGPGSVGGSSSQGGGGGGGVSGGMGSGNGSDDFMTNSVSRDFSIERIIEAEQRAETQCGDRALTFLRVGPYSTVQPDYKGAVSALCQVVNKQLFQMVEYARMMPHFAQVPLDDQVILLKAAWIELLIANVAWCSIVSLDDGGAGGGGGGLGHDGSFERRSPGLQPQQLFLNQSFSYHRNSAIKAGVSAIFDRILSELSVKMKRLNLDRRELSCLKAIILYNPDIRGIKSRAEIEMCREKVYACLDEHCRLEHPGDDGRFAQLLLRLPALRSISLKCQDHLFLFRITSDRPLEELFLEQLEAPPPPGLAMKLE
  
Inhibitor
Name:
BDBM50488454
Synonyms:
CHEMBL2286436
Type:
Small organic molecule
Emp. Form.:
C22H28N2O3
Mol. Mass.:
368.4693
SMILES:
CCOc1ccccc1C(=O)N(NC(=O)c1ccc(CC)cc1)C(C)(C)C
Structure:
Search PDB for entries with ligand similarity: