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Target
Mu-type opioid receptor
Ligand
BDBM50034407
Substrate
n/a
Meas. Tech.
ChEMBL_145425 (CHEMBL747235)
Ki
15±n/a nM
Citation
 Korlipara, VL; Takemori, AE; Portoghese, PS Electrophilic N-benzylnaltrindoles as delta opioid receptor-selective antagonists. J Med Chem 38:1337-43 (1995) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50034407
Synonyms:
1N-{3-[22-cyclopropylmethyl-2,16-dihydroxy-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15,17,19(25)-heptaen-11-ylmethyl]phenyl}-2-bromoacetamide | CHEMBL282518
Type:
Small organic molecule
Emp. Form.:
C35H34BrN3O4
Mol. Mass.:
640.566
SMILES:
Oc1ccc2CC3N(CC4CC4)CCC45[C@@H](Oc1c24)c1c(C[C@@]35O)c2ccccc2n1Cc1cccc(NC(=O)CBr)c1 |TLB:23:22:18.4.5:7.13.12,THB:8:7:22:18.4.5,17:18:22:7.13.12|
Structure:
Search PDB for entries with ligand similarity: