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Target
Cytosol aminopeptidase
Ligand
BDBM50190111
Substrate
n/a
Meas. Tech.
ChEMBL_1821470 (CHEMBL4321130)
Ki
66±n/a nM
Citation
Talma, M; Ma?lanka, M; Mucha, A Recent developments in the synthesis and applications of phosphinic peptide analogs. Bioorg Med Chem Lett 29:1031-1042 (2019) [PubMed] Article
More Info.:
Target
Name:
Cytosol aminopeptidase
Synonyms:
3.4.11.1 | 3.4.11.5 | 3.4.13.23 | AMPL_PIG | Cysteinylglycine-S-conjugate dipeptidase | LAP-3 | LAP3 | Leucine aminopeptidase 3 | Leucyl aminopeptidase | Proline aminopeptidase | Prolyl aminopeptidase
Type:
PROTEIN
Mol. Mass.:
56047.39
Organism:
Sus scrofa
Description:
ChEMBL_101481
Residue:
519
Sequence:
MFLLPLPAAARVAVRQLSVRRFWGPGPDAANMTKGLVLGIYSKEKEDDAPQFTSAGENFDKLVSGKLREILNISGPPLKAGKTRTFYGLHEDFSSVVVVGLGKKGAGVDDQENWHEGKENIRAAVAAGCRQIQDLEIPSVEVDPCGDAQAAAEGAVLGLYEYDELKQKKKVVVSAKLHGSGDQEAWQRGVLFASGQNLARHLMETPANEMTPTRFAEVIEKNLKSASSKTDVHIRPKSWIEEQEMGSFLSVAKGSEEPPVFLEIHYKGSPDASDPPLVFVGKGITFDSGGISIKASANMDLMRADMGGAATICSTIVSAAKLDLPINLVGLAPLCENMPSGKANKPGDVVRAKNGKTIQVDNTDAEGRLILADALCYAHTFNPKVIINAATLTGAMDIALGSGATGVFTNSSWLWNKLFEASIETGDRVWRMPLFEHYTKQIVDCQLADVNNIGKYRSAGACTAAAFLKEFVTHPKWAHLDIAGVMTNKDEVPYLRKGMAGRPTRTLIEFLLRFSQDSA