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Target
Melatonin receptor type 1B
Ligand
BDBM50072658
Substrate
n/a
Meas. Tech.
ChEBML_219514
Ki
40±n/a nM
Citation
 Kloubert, S; Mathé-Allainmat, M; Andrieux, J; Sicsic, S; Langlois, M Synthesis of benzocycloalkane derivatives as new conformationally restricted ligands for melatonin receptors. Bioorg Med Chem Lett 8:3325-30 (1999) [PubMed]  Article 
Target
Name:
Melatonin receptor type 1B
Synonyms:
MEL-1B-R | MTR1B_CHICK | Melatonin | Melatonin receptor | Melatonin receptor type 1B
Type:
Enzyme Catalytic Domain
Mol. Mass.:
33012.73
Organism:
Chick
Description:
Melatonin 0 Chick::P51050
Residue:
289
Sequence:
GNAFVVSLALADLVVALYPYPLVLLAIFHNGWTLGEMHCKVSGFVMGLSVIGSIFNITAIAINRYCYICHSFAYDKVYSCWNTMLYVSLIWVLTVIATVPNFFVGSLKYDPRIYSCTFVQTASSYYTIAVVVIHFIVPITVVSFCYLRIWVLVLQVRRRVKSETKPRLKPSDFRNFLTMFVVFVIFAFCWAPLNFIGLAVAINPSEMAPKVPEWLFIISYFMAYFNSCLNAIIYGLLNQNFRNEYKRILMSLWMPRLFFQDTSKGGTDGQKSKPSPALNNNDQMKTDTL
  
Inhibitor
Name:
BDBM50072658
Synonyms:
CHEMBL114929 | N-(4-Methoxy-bicyclo[4.2.0]octa-1,3,5-trien-7-ylmethyl)-propionamide
Type:
Small organic molecule
Emp. Form.:
C13H17NO2
Mol. Mass.:
219.2796
SMILES:
CCC(=O)NCC1Cc2ccc(OC)cc12
Structure:
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