Reaction Details Report a problem with these data
Target
NF-kappa-B essential modulator
Ligand
BDBM50587700
Substrate
n/a
Meas. Tech.
ChEMBL_2184657 (CHEMBL5096739)
Kd
190±n/a nM
Citation
Hiesinger, K; Dar'in, D; Proschak, E; Krasavin, M Spirocyclic Scaffolds in Medicinal Chemistry. J Med Chem 64:150-183 (2021) [PubMed]
More Info.:
Target
Name:
NF-kappa-B essential modulator
Synonyms:
FIP3 | IKBKG | Inhibitor of NF-kappa-B kinase (IKK) | NEMO | NEMO_HUMAN | NF-kappa-B essential modulator
Type:
PROTEIN
Mol. Mass.:
48190.12
Organism:
Homo sapiens (Human)
Description:
ChEMBL_84013
Residue:
419
Sequence:
MNRHLWKSQLCEMVQPSGGPAADQDVLGEESPLGKPAMLHLPSEQGAPETLQRCLEENQELRDAIRQSNQILRERCEELLHFQASQREEKEFLMCKFQEARKLVERLGLEKLDLKRQKEQALREVEHLKRCQQQMAEDKASVKAQVTSLLGELQESQSRLEAATKECQALEGRARAASEQARQLESEREALQQQHSVQVDQLRMQGQSVEAALRMERQAASEEKRKLAQLQVAYHQLFQEYDNHIKSSVVGSERKRGMQLEDLKQQLQQAEEALVAKQEVIDKLKEEAEQHKIVMETVPVLKAQADIYKADFQAERQAREKLAEKKELLQEQLEQLQREYSKLKASCQESARIEDMRKRHVEVSQAPLPPAPAYLSSPLALPSQRRSPPEEPPDFCCPKCQYQAPDMDTLQIHVMECIE