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Target
Lysophosphatidic acid receptor 3
Ligand
BDBM50166120
Substrate
n/a
Meas. Tech.
ChEMBL_304392 (CHEMBL830042)
EC50
>10000±n/a nM
Citation
 Xu, Y; Aoki, J; Shimizu, K; Umezu-Goto, M; Hama, K; Takanezawa, Y; Yu, S; Mills, GB; Arai, H; Qian, L; Prestwich, GD Structure-activity relationships of fluorinated lysophosphatidic acid analogues. J Med Chem 48:3319-27 (2005) [PubMed]  Article 
Target
Name:
Lysophosphatidic acid receptor 3
Synonyms:
EDG7 | LPA3 | LPAR3 | LPAR3_HUMAN | Lysophosphatidic acid receptor 1/3 | Lysophosphatidic acid receptor 3 (LPAR3) | Lysophosphatidic acid receptor Edg-7
Type:
Enzyme
Mol. Mass.:
40149.72
Organism:
Homo sapiens (Human)
Description:
Q9UBY5
Residue:
353
Sequence:
MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRKFHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNLLVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLAPIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKTVMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDMYGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
  
Inhibitor
Name:
BDBM50166120
Synonyms:
CHEMBL193196 | Hexadecanoic acid (S)-4-fluoro-2-methoxy-4-phosphono-butyl ester
Type:
Small organic molecule
Emp. Form.:
C21H42FO6P
Mol. Mass.:
440.5267
SMILES:
CCCCCCCCCCCCCCCC(=O)OC[C@H](CC(F)P(O)(O)=O)OC
Structure:
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